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Oxymetholone: ​​Ukusetshenziswa, Isikali, Side Effects nokuningi

I-Oxymetholone iyi-synthetic anabolic steroid esetshenziselwa ukwelapha izimo ezithile zezokwelapha. Kuyaziwa ngemiphumela yayo enamandla ekukhuleni kwemisipha kanye nokuzuza kwesisindo. Ekuqaleni ithuthukiswe ngawo-1960, i-Oxymetholone ivame ukunqunywa ezigulini ezinenkinga yokulahlekelwa isisindo ngenxa yezifo ezingapheli, ezifana nomdlavuza noma i-HIV / AIDS. Ibuye isetshenziswe ezimweni ezithile ze-anemia kanye ne-osteoporosis.

⚠️ Ulwazi Lokuphepha Olubalulekile

1. I-Peliosis hepatis: Kuye kwabikwa ukuthi kunezimila ezigcwele igazi esibindini. Lokhu kungase kubonakale njengokungasebenzi kahle kwesibindi okuncane kodwa kungaba yingozi noma kubulale uma ziqhuma.

2. Izimila zesibindi: Kuye kwabikwa kokubili izimila zesibindi ezingengozini (i-hepatic adenoma) kanye nezimila eziyingozi (i-hepatocellular carcinoma). Ukuhoxiswa komuthi kuvame ukuholela ekubuyeleni kwezimila ezingengozini.

3. Izinguquko zamafutha egazini: I-Oxymetholone ibangela ukwehla okuphawulekayo kwe-cholesterol ye-HDL kanye nokwanda kwe-cholesterol ye-LDL, okwandisa kakhulu ingozi ye-atherosclerosis kanye nesifo semithambo yenhliziyo.

Ukukhulelwa: I-Oxymetholone iyi-FDA Pregnancy Category X. Kuyinto kunqatshelwe ngokuphelele ngesikhathi sokukhulelwa ngoba kungabangela ukuvela kwe-virilization yombungu wesifazane, okuhlanganisa nokuvela kwe-virilization yamadoda ngendlela engenakulungiseka.

Ukuvezwa kwe-virilization kwabesifazane: Ukujula kwezwi, i-hirsutism, i-acne, i-clitoromegaly, kanye nokungahambi kahle kokuya esikhathini kungase kwenzeke. Eminye imiphumela, ikakhulukazi ukujula kwezwi, ingase ingabi khona.

Iziguli zezingane: Ukuvalwa kwe-epiphyseal ngaphambi kwesikhathi kungenzeka, okungase kuthinte ukuphakama kokugcina komuntu omdala. Kudingeka ukuqapha ukuvuthwa kwamathambo nge-X-ray njalo ezinyangeni ezi-6.

Ukuqapha: Ukuhlolwa kokusebenza kwesibindi njalo, amaphaneli e-lipid, kanye nokuqapha kwegazi kuyadingeka ngesikhathi sokwelashwa.

Ukusetshenziswa kwe-Oxymetholone

I-Oxymetholone inokusetshenziswa kwezokwelapha okuningana okuvunyelwe, okuhlanganisa:

  1. I-anemia: Isetshenziselwa ukwelapha izinhlobo ezahlukene ze-anemia, ikakhulukazi i-aplastic anemia, lapho umnkantsha wehluleka ukukhiqiza amangqamuzana egazi anele.
  2. Ukukhula Kwesisindo: Inqunyelwe iziguli ezidinga ukuzuza isisindo ngemva kokuhlinzwa, ukulimala, noma ukugula okungapheli.
  3. I-Osteoporosis: Kwezinye izimo, isetshenziselwa ukusiza ukwandisa ukuminyana kwamathambo ezigulini ezine-osteoporosis.
  4. Ukumosha Imisipha: Kuyinzuzo ezigulini ezibhekana nokuwohloka kwemisipha ngenxa yezifo ezingapheli.

Indlela Esebenza

I-Oxymetholone isebenza ngokulingisa imiphumela ye-testosterone emzimbeni. Ibophezela kuma-androgen receptors kumaseli emisipha, ikhuthaza ukuhlanganiswa kwamaprotheni nokugcinwa kwe-nitrogen. Lokhu kuholela ekukhuleni kwemisipha namandla. Ukwengeza, kuthuthukisa ukukhiqizwa kwamangqamuzana egazi abomvu, okuthuthukisa ukulethwa komoya-mpilo emisipha, kuqhubeke nokusekela ukusebenza komzimba nokululama.

Isilinganiso nokuphathwa

Umthamo ojwayelekile we-Oxymetholone uyahlukahluka ngokuya ngesimo sokwelashwa:

  • Abantu abadala: Umthamo wokuqala ojwayelekile ngu-1 kuye ku-5 mg ngekhilogremu ngayinye yesisindo somzimba ngosuku, ngokuvamile ihlukaniswe ngemithamo emibili noma emithathu. Umthamo omkhulu ungakhuphukela ku-150 mg ngosuku, kuye ngokuphendula kwesiguli nokubekezelelana.
  • Iziguli Zezingane: Umthamo wezingane unqunywa umhlinzeki wezempilo ngokusekelwe esisindweni kanye nezidingo ezithile zezokwelapha.

I-Oxymetholone ivame ukulawulwa ngomlomo ngendlela yethebhulethi, ithathwe nokudla ukuze kuncishiswe ukungakhululeki kwamathumbu.

I-Side Effects ye-Oxymetholone

Common side effects of Oxymetholone zihlanganisa:

  • I-nausea
  • Ukuvota
  • Uhudo
  • Ukuphathwa yikhanda
  • Insomnia
  • induna
  • Ukulahlekelwa izinwele

Imiphumela emibi kakhulu ingase ihlanganise:

  • Ukulimala kwesibindi noma izimila
  • Izinkinga zenhliziyo (isb., isifo senhliziyo, isifo sohlangothi)
  • Ukungalingani kweHormonal (isb, i-gynecomastia emadodeni)
  • Ukushintsha kwemizwa, okuhlanganisa ulaka noma ukucindezeleka

Ukusebenzisana kwezidakamizwa

I-Oxymetholone ingaxhumana nemithi eminingi nezinto, kuhlanganise:

  • Ama-anticoagulants (isb., i-warfarin) - angandisa ingozi yokopha.
  • I-insulin kanye nama-oral hypoglycemic agents - angathinta amazinga kashukela egazini.
  • Amanye ama-anabolic steroids - angandisa ingozi yemiphumela emibi.

Ngaso sonke isikhathi wazisa umhlinzeki wakho wokunakekelwa kwezempilo ngayo yonke imithi nezithako zokudla ozithathayo.

Izinzuzo Oxymetholone

Izinzuzo emitholampilo usebenzisa Oxymetholone zihlanganisa:

  • Ukuzuza Okusheshayo Kwemisipha: Ingenye ye-steroids ephumelela kakhulu yokwandisa isisindo semisipha ngokushesha.
  • Ukubuyisela Okuthuthukisiwe: Isiza ekululameni ngokushesha ekulimaleni nasekuhlinzweni.
  • Ukusebenza Okuthuthukisiwe: Abasubathi bangase babe namandla athuthukisiwe nokukhuthazela.
  • Ukukhiqizwa Kwamaseli Abomvu Egazi Okunyusiwe: Lokhu kungaholela ku-oxygenation engcono yemisipha, kuthuthukise ukusebenza komzimba jikelele.

Contraindications of Oxymetholone

Abantu abathile kufanele bakugweme ukusebenzisa i-Oxymetholone, okuhlanganisa:

  • Abesifazane abakhulelwe noma abancelisayo, njengoba kungalimaza umbungu noma usana.
  • Iziguli ezinesifo sesibindi noma izimila zesibindi.
  • Abantu abanomdlavuza wendlala yesinye noma umdlavuza webele emadodeni.
  • Labo abanomlando wesifo senhliziyo noma unhlangothi.

Ukuqapha Nezexwayiso

Ngaphambi kokuqala i-Oxymetholone, iziguli kufanele zihlolwe zelebhu ethize ukuze zihlole ukusebenza kwesibindi kanye nempilo yonke. Kubalulekile ukuqapha noma yiziphi izimpawu zokulimala kwesibindi noma ukungalingani kwe-hormonal ngesikhathi sokwelashwa. Iziguli kufanele futhi zixoxe ngomlando wazo wezokwelapha ophelele nomhlinzeki wazo wokunakekelwa kwezempilo ukuze kuqinisekiswe ukuphepha.

Imibuzo Evame Ukubuzwa

  1. I-Oxymetholone isetshenziselwa ini?
    I-Oxymetholone isetshenziselwa ukwelapha i-anemia, ukukhuthaza ukuzuza kwesisindo ezigulini ezilulama ekuguleni, nokuthuthukisa ukuminyana kwamathambo e-osteoporosis.
  2. Kufanele ngithathe kanjani i-Oxymetholone?
    Ithathwa ngomlomo, ngokuvamile ngokudla, ukunciphisa ukucasuka kwesisu. Landela imiyalelo kadokotela wakho mayelana nomthamo.
  3. Yimiphi imiphumela emibi evamile?
    Imiphumela emibi evamile ihlanganisa isicanucanu, ubuhlungu bekhanda, nezinduna. Imiphumela emibi kakhulu ingabandakanya ukulimala kwesibindi kanye nezinkinga zenhliziyo.
  4. Ingabe abesifazane bangasebenzisa i-Oxymetholone?
    Yebo, kodwa kufanele baqaphele ngenxa yengozi ye-virilization (ukuthuthukiswa kwezici zesilisa).
  5. Ingabe i-Oxymetholone iphephile ukusetshenziswa isikhathi eside?
    Ukusetshenziswa isikhathi eside kungaholela emiphumeleni emibi kakhulu, ngakho kufanele iqashwe eduze ngumhlinzeki wezempilo.
  6. Yini okufanele ngiyenze uma ngiphuthelwa umthamo?
    Thatha umthamo ogejiwe ngokushesha nje lapho ukhumbula. Uma kuseduze nomthamo olandelayo, yeqa umthamo futhi uqalise kabusha isimiso sakho esivamile.
  7. Ngingakwazi ukuphuza utshwala ngenkathi ngithatha i-Oxymetholone?
    Kunconywa ukugwema utshwala, njengoba kungandisa ingozi yokulimala kwesibindi.
  8. I-Oxymetholone iwuthinta kanjani umoya wami?
    Abanye abasebenzisi bangase babe nokushintshashintsha kwemizwa, ulaka, noma ukucindezeleka. Bika noma yiziphi izinguquko ezibalulekile kudokotela wakho.
  9. Ngingakwazi ukusebenzisa i-Oxymetholone ekwakheni umzimba?
    Nakuba ngezinye izikhathi isetshenziswa kabi ekwakheni umzimba, kubalulekile ukuyisebenzisa ngaphansi kokuqondisa kwezokwelapha ngenxa yezingozi zempilo ezingaba khona.
  10. Yini okufanele ngiyenze uma ngiba nemiphumela emibi kakhulu?
    Funa usizo lwezokwelapha ngokushesha uma uhlangabezana nemiphumela emibi kakhulu njengobuhlungu besifuba, i-jaundice, noma izinguquko ezinzima zemizwa.

Amagama Omkhiqizo

I-Oxymetholone itholakala ngaphansi kwamagama amaningana emikhiqizo, okuhlanganisa:

  • Anadrol
  • I-Oxydrolone
  • I-Anapolon

Isiphetho

I-Oxymetholone iyi-steroid enamandla ye-anabolic enezicelo ezithile zezokwelapha, ikakhulukazi ekwelapheni i-anemia nokukhuthaza ukukhuluphala. Nakuba inikeza izinzuzo ezibalulekile, futhi iza nemiphumela engemihle engaba khona kanye nezingozi. Kubalulekile ukusebenzisa lo muthi ngaphansi kokuqondisa kochwepheshe bezempilo ukuze uqinisekise ukuphepha nokusebenza ngempumelelo.

Umshwana wokuzihlangula: Lolu lwazi lwenzelwe izinjongo zokufundisa kuphela futhi aluthatheli indawo iseluleko sochwepheshe bezokwelapha. Hlala uthintana nodokotela wakho mayelana nezinkinga zezokwelapha.

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